#0132: Aryl and Vinyl Amination
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TECH FIELD(S)
Research Tool
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FEATURES
The invention provides methodology for carbon-nitrogen bond formation via vinyl or aryl amination. An sp2 hybridized radical is reacted with an azomethine moiety to form pyrrolidine and indole compounds.
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BENEFITS
The invention provides a facile process for the syntheis of compunds having the pyrrolidine or indole subunit and is especially advantageous for compounds having acid or base labile functional groups and/or is comprised of chiral centers susceptible to acid/base epimerization.
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INVENTOR(S)
Jeffrey N. Johnston and Rajesh Viswanathan
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INTELLECTUAL PROPERTY STATUS
US 6,670,479 and US 7,078,567
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CONTACT INFORMATION
For additional information on this technology, please contact Bill Brizzard, Director of Technology Transfer , IURTC:
Indiana University Research & Technology Corporation
501 North Morton Street, Suite 204
Bloomington, IN 47404
Telephone:812-855-3597
bbrizzar@iu.edu
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